BDBM501744 N-Cyclopentyl-3-(5-((7-methyl-5-(2-(4-methylpiperazin-1-yl)ethoxy)-9-oxo-9H-xanthen-3-yl)oxy)pyridin-2-yl)propanamide::US11028064, Example 58

SMILES CN1CCN(CCOc2cc(C)cc3c2oc2cc(Oc4ccc(CCC(=O)NC5CCCC5)nc4)ccc2c3=O)CC1

InChI Key InChIKey=VJZKCRBDGMLOQY-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 501744   

TargetVascular endothelial growth factor receptor 2(Homo sapiens (Human))
Auckland Uniservices

US Patent
LigandPNGBDBM501744(N-Cyclopentyl-3-(5-((7-methyl-5-(2-(4-methylpipera...)
Affinity DataIC50: >1.00E+4nMAssay Description:IC50 values were determined using the Z′-LYTEŽ activity assay, with ATP concentration used at Km app for the specific assay (500 μM ATP fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent
TargetMacrophage colony-stimulating factor 1 receptor(Homo sapiens (Human))
Auckland Uniservices

US Patent
LigandPNGBDBM501744(N-Cyclopentyl-3-(5-((7-methyl-5-(2-(4-methylpipera...)
Affinity DataIC50: <100nMAssay Description:IC50 values were determined using the Z′-LYTEŽ activity assay, with ATP concentration used at Km app for the specific assay (500 μM ATP fo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent