BDBM501840 4-{2-(4-methoxyphenyl)-1- methyl-5-[4- (methylamino)piperidyl]-6-oxo-3- hydropyridyl}benzenecarbonitrile::US11028066, Example 78
SMILES CNC1CCN(CC1)c1cc(-c2ccc(cc2)C#N)c(-c2ccc(OC)cc2)n(C)c1=O
InChI Key InChIKey=VOJZLWHSUQQPHK-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 501840
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Celgene Quanticel Research
US Patent
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of LSD1 activity is based on Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The inhibitory properties ...More data for this Ligand-Target Pair