BDBM501845 4-[5-(4-aminopiperidin-1-yl)-2-(3- fluoro-4-methoxyphenyl)-1- methyl-6-oxopyridin-3- yl]benzonitrile::US11028066, Example 83
SMILES COc1ccc(cc1F)-c1c(cc(N2CCC(N)CC2)c(=O)n1C)-c1ccc(cc1)C#N
InChI Key InChIKey=QFTURYYVMWHLTJ-UHFFFAOYSA-N
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 501845
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Celgene Quanticel Research
US Patent
Celgene Quanticel Research
US Patent
Affinity DataIC50: <100nMAssay Description:The enzymatic assay of LSD1 activity is based on Time Resolved-Fluorescence Resonance Energy Transfer (TR-FRET) detection. The inhibitory properties ...More data for this Ligand-Target Pair