BDBM50185473 4-(3-(4-chlorophenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]octan-8-yl)-1-(4-fluorophenyl)butan-1-one::4-[3-(4-Chloro-phenyl)-3-hydroxy-8-aza-bicyclo[3.2.1]oct-8-yl]-1-(4-fluoro-phenyl)-butan-1-one::4-[3-(4-Chlorophenyl)-3-hydroxy-8-azabicyclo[3.2.1]oct-8-yl]-1-(4-fluorophenyl)butan-1-one::CHEMBL210578
SMILES OC1(CC2CCC(C1)N2CCCC(=O)c1ccc(F)cc1)c1ccc(Cl)cc1
InChI Key InChIKey=CXQUOFVDYCOSEZ-UHFFFAOYSA-N
Data 35 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 35 hits for monomerid = 50185473
Affinity DataKi: 0.309nMAssay Description:Cataleptogenic effect against cloned human Dopamine receptor D2 in male Sprague-Dawley rats in a bar testMore data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:In vitro ability to inhibit the binding of [3H]-spiperone to cloned human Dopamine receptor D2 using apomorphine induced climbing test in male Swiss ...More data for this Ligand-Target Pair
Affinity DataKi: 0.310nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 0.708nMAssay Description:Cataleptogenic effect against cloned human Dopamine receptor D3 in male Sprague-Dawley rats in a bar testMore data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:In vitro ability to inhibit the binding of [3H]-7-OH-DPAT to cloned human Dopamine receptor D3 using apomorphine induced climbing test in male Swiss ...More data for this Ligand-Target Pair
Affinity DataKi: 0.710nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human cloned dopamine D2 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human cloned dopamine D2 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D2 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D3 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to dopamine D3 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Binding affinity to human cloned dopamine D3 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Displacement of [125I]DOI from human dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity to human cloned dopamine D4 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 5.30nMAssay Description:Binding affinity to human cloned dopamine D4.4 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Displacement of [3H]N-methylspiperone from rat dopamine D4 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:In vitro ability to inhibit the binding of [3H]-spiperone to cloned human dopamine receptor D4 using apomorphine induced climbing test in male Swiss ...More data for this Ligand-Target Pair
Affinity DataKi: 12nMAssay Description:Cataleptogenic effect against cloned human dopamine receptor D4 in male Sprague-Dawley rats in a bar testMore data for this Ligand-Target Pair
Affinity DataKi: 27.7nMAssay Description:Binding affinity to human cloned 5HT1A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Binding affinity to human cloned 5HT1A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 28nMAssay Description:Displacement of [3H] 8-OH-DPAT from human 5-HT1A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 30.9nMAssay Description:Binding affinity to human cloned 5HT2A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Displacement of [3H]Ketanserin from human 5-HT2A receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 31nMAssay Description:Binding affinity to human cloned 5HT2A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 39nMAssay Description:Binding affinity to human cloned adrenergic alpha-1A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 43nMAssay Description:Binding affinity to human cloned adrenergic alpha-1B receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 143nMAssay Description:Binding affinity to human cloned adrenergic alpha-2C receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 516nMAssay Description:Binding affinity to human cloned adrenergic alpha-2B receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 872nMAssay Description:Binding affinity to human cloned 5HT2C receptor by radioligand binding assayMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2C(Rattus norvegicus (Rat))
Florida A&M University
Curated by ChEMBL
Florida A&M University
Curated by ChEMBL
Affinity DataKi: 872nMAssay Description:Displacement of [3H]Mesulergine from rat 5-HT2C receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 872nMAssay Description:Binding affinity to human cloned 5HT2C receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.84E+3nMAssay Description:Binding affinity to human cloned adrenergic alpha-2A receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.78E+3nMAssay Description:Displacement of [3H]Pyrilamine from human histamine H1 receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.78E+3nMAssay Description:Binding affinity to human cloned histamine H1 receptor by radioligand binding assayMore data for this Ligand-Target Pair
Affinity DataKi: 8.78E+3nMAssay Description:Binding affinity to human cloned histamine H1 receptorMore data for this Ligand-Target Pair