BDBM501872 US11028075, Example 5
SMILES CN(C)[C@H]1C[C@H](CC[C@@H]1Nc1cc(F)c(cc1OC(F)F)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F
InChI Key InChIKey=CPGVCENSNKQVCS-LRQRDZAKSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 501872
Affinity DataIC50: 0.519nMAssay Description:The following voltage clamp electrophysiology studies are performed on representative compounds using cells heterologously expressing Nav1.7 or Nav1....More data for this Ligand-Target Pair
Affinity DataIC50: 1.37nMAssay Description:Saturation experiments. A competitive NaV1.7 inhibitor having a methyl group is tritiated. Three tritiums are incorporated in place of methyl hydroge...More data for this Ligand-Target Pair