BDBM501922 US11028075, Example 55
SMILES CN(C)[C@H]1C[C@H](CC[C@@H]1N1C(=O)CCc2cc(c(F)cc12)S(=O)(=O)Nc1ccncn1)c1cccc(c1)C(F)(F)F
InChI Key InChIKey=JXCCMRIQEWZXQL-OEOAZWSVSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 501922
Affinity DataIC50: 2.68nMAssay Description:The following voltage clamp electrophysiology studies are performed on representative compounds using cells heterologously expressing Nav1.7 or Nav1....More data for this Ligand-Target Pair
Affinity DataIC50: 6.73nMAssay Description:Saturation experiments. A competitive NaV1.7 inhibitor having a methyl group is tritiated. Three tritiums are incorporated in place of methyl hydroge...More data for this Ligand-Target Pair