BDBM50236543 CHEMBL4078550
SMILES CC(=O)Nc1ccc(cc1)-c1cnc2[nH]cc(-c3ccc(O)cc3)c2c1
InChI Key InChIKey=PVFNDFZQGWYILU-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50236543
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1A(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 6.60nMAssay Description:Inhibition of DYRK1A (unknown origin) using woodtide as substrate after 10 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 1B(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 38nMAssay Description:Inhibition of DYRK1B (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity tyrosine-phosphorylation-regulated kinase 2(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataIC50: 536nMAssay Description:Inhibition of DYRK2 (unknown origin) using woodtide as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair
TargetDual specificity protein kinase CLK1(Homo sapiens (Human))
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Qimr Berghofer Medical Research Institute
Curated by ChEMBL
Affinity DataEC50: 3.50E+4nMAssay Description:Inhibition of CLK1 (unknown origin) using KKGRSRSRSRSRSR as substrate after 40 mins in presence of [gamma-33P]ATP by microbeta scintillation countingMore data for this Ligand-Target Pair