BDBM50238256 CHEMBL4078384

SMILES COc1ccc(CCc2nc3cc(ccc3n2CCN2CCOCC2)-c2c(C)noc2C)cc1OC

InChI Key InChIKey=JKZPYPCQYQOWSK-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50238256   

TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238256(CHEMBL4078384)
Affinity DataIC50:  470nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238256(CHEMBL4078384)
Affinity DataIC50:  9.40E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed