BDBM50238258 CHEMBL4075476

SMILES COc1cccc(CCc2nc3cc(ccc3n2CCN2CCOCC2)-c2c(C)noc2C)c1

InChI Key InChIKey=OQALUPRPYHSUER-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50238258   

TargetCREB-binding protein(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238258(CHEMBL4075476)
Affinity DataIC50:  310nMAssay Description:Inhibition of CREBBP (unknown origin) by FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBromodomain-containing protein 4(Homo sapiens (Human))
Pfizer

Curated by ChEMBL
LigandPNGBDBM50238258(CHEMBL4075476)
Affinity DataIC50:  4.60E+3nMAssay Description:Inhibition of BRD4 (unknown origin) by fluorescence polarization assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed