BDBM50274739 CHEMBL4127485
SMILES COc1ccc(C[C@H](NC(=O)[C@@H](CCCNC(N)=N)NC(=O)[C@@H](N)Cc2c(C)cc(O)cc2C)C(=O)NCC(N)=O)cc1
InChI Key InChIKey=UAJIBHYIOKBSNN-VXNXHJTFSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50274739
Affinity DataIC50: 0.901nMAssay Description:Agonist activity at mu-opioid receptor in guinea pig ileum assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair
Affinity DataIC50: 0.470nMAssay Description:Displacement of [125I]-DAMGO from mouse Flag-tagged mu-opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 70nMAssay Description:Displacement of [125I]-Deltorphin 2 from mouse Flag-tagged delta-opioid receptor expressed in HEK293 cell membranes after 60 mins by gamma countingMore data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Agonist activity at delta-opioid receptor in mouse vasa deferens assessed as inhibition of electrically induced contractionsMore data for this Ligand-Target Pair