BDBM50277339 2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfonyl)phenyl)cyclopropanecarboxamide::CHEMBL472856

SMILES Cc1ccc(NC(=O)C2C(C)(C)C2(C)C)cc1S(=O)(=O)N1CCOCC1

InChI Key InChIKey=JUQFVKJYAGSDTL-UHFFFAOYSA-N

Data  6 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 8 hits for monomerid = 50277339   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP 55940 from human CB2 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP55940 from human cloned CB2 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  23nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]CP55940 from human cloned CB1 receptor by scintillation spectrometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataKi:  3.40E+3nMAssay Description:Displacement of [3H]CP 55940 from human CB1 receptor in cell free systemMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Adolor

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at rat brain CB2 receptor by GTPgammaS binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50277339(2,2,3,3-tetramethyl-N-(4-methyl-3-(morpholinosulfo...)
Affinity DataEC50:  11nMAssay Description:Agonist activity at human cloned CB2 receptor assessed as stimulation of [35S]GTPgammaS bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed