BDBM50287703 (E)-1-[(S)-2-(2-Hydroxy-ethyl)-piperidin-1-yl]-3-(2-phenyl-pyrazolo[1,5-a]pyridin-3-yl)-propenone::CHEMBL61845
SMILES OCC[C@@H]1CCCCN1C(=O)\C=C\c1c(nn2ccccc12)-c1ccccc1
InChI Key InChIKey=OPLOPFHUHFGKMJ-HYSAVQALSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50287703
Affinity DataIC50: 1.13E+4nMAssay Description:Inhibition of [3H]NECA specific binding against Adenosine A2 receptors of rat striatal membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 17nMAssay Description:Inhibition of [3H]-CHA binding against Adenosine A1 receptors of rat cortical membranesMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Inhibition of adenosine induced negative inotropic activity against guinea-pig atria (Adenosine A1 receptor)More data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Compound was evaluated for inhibition of adenosine induced relaxation against guinea-pig aorta (Adenosine A2 receptor).More data for this Ligand-Target Pair