BDBM50303776 CHEMBL568525::N-((6S,9S,12S)-1,17-diamino-6-(4-carbamimidoylbenzylcarbamoyl)-1,17-diimino-9-isopropyl-8,11-dioxo-2,7,10,16-tetraazaheptadecan-12-yl)decanamide
SMILES [#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6]-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6@@H](-[#6](-[#6])-[#6])-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](/[#7])-[#7])-[#6](=O)-[#7]-[#6]-c1ccc(cc1)-[#6](-[#7])=[#7]
InChI Key InChIKey=QMAXHSLPLMYIPN-YCVJPRETSA-N
Data 6 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50303776
Affinity DataKi: 1.60nMAssay Description:Inhibition of human furin by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 6(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 3nMAssay Description:Inhibition of human PACE4 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 3.70nMAssay Description:Inhibition of human PC1/3 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 5(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 6.30nMAssay Description:Inhibition of human PC5/6 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
Affinity DataKi: 55nMAssay Description:Inhibition of human PC2 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair
TargetProprotein convertase subtilisin/kexin type 7(Homo sapiens (Human))
Philipps University Marburg
Curated by ChEMBL
Philipps University Marburg
Curated by ChEMBL
Affinity DataKi: 968nMAssay Description:Inhibition of human PC7 expressed in Drosophila schneider 2 cells by fluorescence assayMore data for this Ligand-Target Pair