BDBM50341559 7-chloro-3-(3,5-dimethylphenyl)-4-(2-(piperidin-2-yl)ethoxy)-6-(pyrimidin-4-yl)quinolin-2(1H)-one::CHEMBL1766106
SMILES Cc1cc(C)cc(c1)-c1c(OCCC2CCCCN2)c2cc(c(Cl)cc2[nH]c1=O)-c1ccncn1
InChI Key InChIKey=YAWOHPIYLYGVRK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50341559
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataKi: 1.40E+3nMAssay Description:Displacement of I125-somatostatin-14 from human SST2 expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Merck Research Laboratories
Curated by ChEMBL
Merck Research Laboratories
Curated by ChEMBL
Affinity DataIC50: 3.20nMAssay Description:Antagonist activity at GnRH receptor by GnRHMore data for this Ligand-Target Pair