BDBM50341563 7-chloro-3-(3,5-dimethylphenyl)-6-phenyl-4-(2-(piperidin-2-yl)ethoxy)-1,2-dihydroquinoline::CHEMBL1766110

SMILES Cc1cc(C)cc(c1)C1=C(OCCC2CCCCN2)c2cc(c(Cl)cc2NC1)-c1ccccc1

InChI Key InChIKey=MRYYDCIBVWPZNW-UHFFFAOYSA-N

Data  1 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50341563   

TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50341563(7-chloro-3-(3,5-dimethylphenyl)-6-phenyl-4-(2-(pip...)
Affinity DataKi:  0.180nMAssay Description:Displacement of I125-somatostatin-14 from human SST2 expressed in CHO cells after 3 hrs by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50341563(7-chloro-3-(3,5-dimethylphenyl)-6-phenyl-4-(2-(pip...)
Affinity DataIC50:  7.60nMAssay Description:Agonist activity at human SST2 expressed in CHO cells assessed as inhibition of forskolin-stimulated cAMP release after 40 mins by luminescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed