BDBM50355909 CHEMBL1910195

SMILES Oc1ccc(cc1)-c1cncc(c1)-c1cc2ccc(O)cc2[nH]1

InChI Key InChIKey=BKQKPRMOYMYOAI-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50355909   

LigandPNGBDBM50355909(CHEMBL1910195)
Affinity DataIC50:  60nMAssay Description:Inhibition of rat recombinant GST-fused DYRK1A expressed in Escherichia coli using myelin protein and [33P-gamma]-ATP after 30 mins by scintillation ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCyclin-dependent kinase 5 activator 1(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50355909(CHEMBL1910195)
Affinity DataIC50:  160nMAssay Description:Inhibition of human recombinant CDK5/p25 using histone H1 and [33P-gamma]-ATP after 30 mins by scintillation countingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Sus scrofa)
Universit£

Curated by ChEMBL
LigandPNGBDBM50355909(CHEMBL1910195)
Affinity DataIC50:  1.10E+3nMAssay Description:Inhibition of porcine brain GSK3-beta assessed as incorporation of [gamma-33P]-ATP into YRRAAVPPSPSLSRHSSPHQSpEDEEE substrate after 30 mins by scinti...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed