BDBM50410544 CHEMBL390519
SMILES OC(=O)c1cccc(NC(=O)c2[nH]c(nc2COC23CC4CC(CC(C4)C2)C3)C2CCCCC2)c1
InChI Key InChIKey=RKPUHYCGNGSOCF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50410544
Affinity DataKi: 11nMAssay Description:Displacement of [125I]BH-CCK8-8S from CCK2 receptor in canine gastric mucosaChecked by AuthorMore data for this Ligand-Target Pair
TargetGastrin/cholecystokinin type B receptor(Homo sapiens (Human))
James Black Foundation
Curated by ChEMBL
James Black Foundation
Curated by ChEMBL
Affinity DataKi: 19nMAssay Description:Displacement of [3H]BH-CCK-8S from human recombinant CCK2 receptor expressed in NIH3T3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataKi: 501nMAssay Description:Displacement of [125I]BH-CCK-8S from CC1 receptor expressed in guinea pig pancreatic cellsMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:Displacement of [3H]L-364718 from human recombinant CCK1 receptor expressed in PC3 cellsChecked by AuthorMore data for this Ligand-Target Pair
Affinity DataIC50: 19nMAssay Description:Concentration required to inhibit the binding of [125I]-BH-CCK-8S radioligand to canine gastric mucosa CCK2 receptorMore data for this Ligand-Target Pair