BDBM50413761 CHEMBL390094
SMILES CC(C)[C@H](NC(=O)[C@@H]1CSSC(C)(C)[C@@H](NC(=O)[C@@H](N)CC(O)=O)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N1)C(O)=O
InChI Key InChIKey=IWPZSQYTMKMNRX-POSKKVNKSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50413761
Affinity DataKi: 0.200nMAssay Description:Ability to displace radioligand [125I]Tyr-hU-II from human recombinant Urotensin 2 receptor in CHO-K1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Binding affinity towards human Urotensin 2 receptor was determinedMore data for this Ligand-Target Pair
Affinity DataKi: 0.200nMAssay Description:Displacement of [125I]urotensin-2 from human UT2 receptor expressed in CHO-K1 cells by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataEC50: 0.251nMAssay Description:Agonist activity at UT2 receptor in Albino rat aorta assessed as induction of aortic contractionMore data for this Ligand-Target Pair