BDBM50420542 CHEMBL2086965
SMILES Oc1ccc(Br)cc1\C=N\NC(=O)c1cc2ccccc2cc1O
InChI Key InChIKey=XTFYZTFVHVNUEN-KEBDBYFISA-N
Data 5 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50420542
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled SRC1-4 from dexamethasone-GR complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERalpha complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.33E+4nMAssay Description:Antagonist activity at wild type AR LBD assessed as inhibition of DHT-induced fluorescent labeled D11-FxxLF recruitment after 2 to 4 hrs by TR-FRET a...More data for this Ligand-Target Pair
Affinity DataIC50: 2.25E+4nMAssay Description:Antagonist activity at PR assessed as inhibition of progesterone-induced fluorescent labelled SRC1-4 recruitment after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: >1.00E+5nMAssay Description:Displacement of fluorescent labelled PGC-1alpha from estradiol-ERbeta complex after 2 to 4 hrs by TR-FRET assayMore data for this Ligand-Target Pair