BDBM50425662 CHEMBL2315528
SMILES OC(=O)CCc1ccc(cc1)C#Cc1ccccc1CC#N
InChI Key InChIKey=AMKACOPNIVQTHQ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50425662
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataKi: 204nMAssay Description:Displacement of 3-(2-Fluoro-4-((2'-methyl-4'-(2-(2-((7-nitrobenzo[c][1,2,5]-oxadiazol-4-yl)amino)ethoxy)ethoxy)-[1,1'-biphenyl]-3-yl)-methoxy)phenyl)...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 4(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 776nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA4 receptor transfected in HEK293 cells after 5 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human FFA1 assessed as calcium mobilization measured for 50 intervals of 0.4 secs by microplate reader analysisMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 69nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA1 receptor transfected in HEK293 cells after 5 mins by BRET assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 20nMAssay Description:Agonist activity at human FFA1 receptor transfected in human 1321N1 cells by calcium mobilization assayMore data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 62nMAssay Description:Agonist activity at human C-terminal eYFP-tagged FFA1 receptor expressed in HEK-293 cells assessed as beta-arrestin2 recruitment incubated for 5 mins...More data for this Ligand-Target Pair
TargetFree fatty acid receptor 1(Homo sapiens (Human))
University Of Southern Denmark
Curated by ChEMBL
University Of Southern Denmark
Curated by ChEMBL
Affinity DataEC50: 240nMAssay Description:Agonist activity at C-terminal yellow fluorescent protein-fused human FFA1 receptor transfected in HEK293 cells after 5 mins by BRET assay in presenc...More data for this Ligand-Target Pair