BDBM506429 US11045457, Example 29
SMILES CN1C[C@@H](NC(=O)C(C)(C)COc2ncccc2OC(F)(F)F)[C@@H](C1)c1cn(C)nc1C
InChI Key InChIKey=HCQKSFFXWPTXIQ-JKSUJKDBSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 506429
Affinity DataEC50: 3.98nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
Affinity DataIC50: 398nMAssay Description:This membrane-based assay measures the ability of compounds to competitively inhibit binding of I-125 labeled somatostatin to SSTR1 in membranes from...More data for this Ligand-Target Pair
Affinity DataIC50: 39.8nMAssay Description:This membrane-based assay measures the ability of compounds to competitively inhibit binding of I-125 labeled somatostatin to SSTR4 in membranes from...More data for this Ligand-Target Pair