BDBM506539 US11045457, Example 139::US11045457, Example 177
SMILES C[C@@H]1C[C@H](CCN1C)NC(=O)C(C)(C)COc1ncccc1C(F)(F)F
InChI Key InChIKey=PAZHTQRFSKYTCX-OLZOCXBDSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 506539
Affinity DataEC50: 12.6nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
Affinity DataEC50: 126nMAssay Description:This cell-based assay measures the ability of compounds to inhibit forskolin stimulated cAMP in CHO-K1 cells overexpressing SSTR4. CHO-K1 cells overe...More data for this Ligand-Target Pair
Affinity DataIC50: 6.31E+3nMAssay Description:This membrane-based assay measures the ability of compounds to competitively inhibit binding of I-125 labeled somatostatin to SSTR1 in membranes from...More data for this Ligand-Target Pair
Affinity DataIC50: 63.1nMAssay Description:This membrane-based assay measures the ability of compounds to competitively inhibit binding of I-125 labeled somatostatin to SSTR4 in membranes from...More data for this Ligand-Target Pair