BDBM508622 (R or S)-8-[2-(6,6-difluoro-2- azabicyclo[2.2.1]hept-2-yl)ethyl]-2,2- difluoro[1,3]dioxolo[4,5-h][1,2,4] triazolo[1,5-c]quinazolin-5-amine (faster eluting b)::US11046714, Example 66::US11046714, Example 67
SMILES Nc1nc2c3OC(F)(F)Oc3ccc2c2nc(CCN3CC4CC3C(F)(F)C4)nn12
InChI Key InChIKey=KHYQDCRSZOBGGT-UHFFFAOYSA-N
Data 2 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 508622
Affinity DataKi: 3nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair
Affinity DataKi: 3.5nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair