BDBM508712 (R or S)-2,2-difluoro-8-(1-pyrimidin- 5-ylpiperidin-3-yl)[1,3]dioxolo[4,5- h][1,2,4]triazolo[1,5-c]quinazolin-5- amine (faster eluting b)::US11046714, Example 146
SMILES Nc1nc2c3OC(F)(F)Oc3ccc2c2nc(nn12)[C@H]1CCCN(C1)c1cncnc1
InChI Key InChIKey=JJESMNPJLANBMC-JTQLQIEISA-N
Data 1 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 508712
Affinity DataKi: 44nMAssay Description:The following table shows representative data for the compounds of the Examples as A2a receptor antagonists as determined by a competition binding as...More data for this Ligand-Target Pair