BDBM534178 6-Cyclopropyl-N-(2-ethoxyphenyl)sulfonyl-4-(trifluoromethyl)benzofuran-2-carboxamide::WO2022081842, Example 51

SMILES CCOc1ccccc1S(=O)(=O)NC(=O)c1cc2c(cc(cc2o1)C1CC1)C(F)(F)F

InChI Key InChIKey=IXBLCUJEGKCDGV-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534178   

TargetHistone acetyltransferase KAT6A [507-778](Homo sapiens)
The Broad Institute

WIPO
LigandPNGBDBM534178(6-Cyclopropyl-N-(2-ethoxyphenyl)sulfonyl-4-(triflu...)
Affinity DataIC50:  26nMAssay Description: Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed