BDBM534180 6-Cyclopropyl-N-(2-phenylphenyl)sulfonyl-4-(trifluoromethyl)benzofuran-2-carboxamide::WO2022081842, Example 53

SMILES FC(F)(F)c1cc(cc2oc(cc12)C(=O)NS(=O)(=O)c1ccccc1-c1ccccc1)C1CC1

InChI Key InChIKey=OQXDTIGBFBGVCP-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 534180   

TargetHistone acetyltransferase KAT6A [507-778](Homo sapiens)
The Broad Institute

WIPO
LigandPNGBDBM534180(6-Cyclopropyl-N-(2-phenylphenyl)sulfonyl-4-(triflu...)
Affinity DataIC50:  43nMAssay Description: Kat6a inhibitory activities of the compounds described in the present invention were quantified using a Fluorescence Resonance Energy Transfer (TR-F...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed