BDBM82547 SRIF-D-Trp8
SMILES C[C@@H](O)[C@@H]1NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@@H](NC(=O)[C@H](CCCCN)NC(=O)[C@@H](Cc2c[nH]c3ccccc23)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](Cc2ccccc2)NC(=O)[C@H](CC(N)=O)NC(=O)[C@H](CCCCN)NC(=O)[C@H](CSSC[C@H](NC(=O)[C@H](CO)NC1=O)C(O)=O)NC(=O)CNC(=O)[C@H](C)N)[C@@H](C)O
InChI Key InChIKey=NHXLMOGPVYXJNR-ZPHDWPCDSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 13 hits for monomerid = 82547
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.00100nMAssay Description:Displacement of [125I]-somatostatin from human SSTR2 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.320nMAssay Description:Displacement of [125I]-somatostatin from human SSTR1 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataKi: 0.460nMAssay Description:Displacement of [125I]-somatostatin from human SSTR5 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 0.610nMAssay Description:Displacement of [125I]-somatostatin from human SSTR3 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataKi: 5.80nMAssay Description:Displacement of [125I]-somatostatin from human SSTR4 expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataIC50: 1.10nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst2 receptor in CCL39 cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataEC50: 0.630nMAssay Description:Agonist activity at human sst3 receptor expressed in CCL39 cells after 5 hrs by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataIC50: 3.10nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst5 receptor in HEK293 cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataIC50: 2.30nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst4 receptor in CCL39 cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
University Of Toronto
Curated by PDSP Ki Database
University Of Toronto
Curated by PDSP Ki Database
Affinity DataIC50: 2.40nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst3 receptor in CCL39 cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Institute For Research In Biomedicine (Irb Barcelona)
Curated by ChEMBL
Affinity DataIC50: 2.30nMAssay Description:Displacement of 125I-[LTT]-SRIF-28 from human sst1 receptor in CHO cells after 2 hrs by autoradiographyMore data for this Ligand-Target Pair