BDBM86428 SB-258585
SMILES COc1ccc(NS(=O)(=O)c2ccc(I)cc2)cc1N1CCN(C)CC1
InChI Key InChIKey=BDHMSYNBSBZCAF-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 86428
Affinity DataKi: 0.75nMAssay Description:Antagonist activity at mouse wild type 5HT6 receptor expressed in COS7 cells assessed as inhibition of seratonin-induced cAMP accumulation by HTRF as...More data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline
Curated by PDSP Ki Database
Glaxosmithkline
Curated by PDSP Ki Database
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline
Curated by PDSP Ki Database
Glaxosmithkline
Curated by PDSP Ki Database
Affinity DataKi: 2.5nMAssay Description:Binding affinity for human 5-hydroxytryptamine 6 receptorChecked by AuthorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Glaxosmithkline
Curated by PDSP Ki Database
Glaxosmithkline
Curated by PDSP Ki Database
Affinity DataIC50: 19nMAssay Description:Antagonist activity at human 5-HT6 receptor expressed in human HeLa cells assessed as inhibition of 5-HT-induced cAMP accumulation pretreated for 10 ...More data for this Ligand-Target Pair