BDBM93410 PHD Inhibitor, 5

SMILES CC(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1

InChI Key InChIKey=NGUVRCCRQHFTMR-UHFFFAOYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 93410   

TargetEgl nine homolog 1(Homo sapiens (Human))
Amgen Inc

LigandPNGBDBM93410(PHD Inhibitor, 5)
Show SMILES CC(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1
Show InChI InChI=1S/C16H17N3O6/c1-8(20)17-6-9-3-4-11-10(5-9)14(23)13(16(25)19(11)2)15(24)18-7-12(21)22/h3-5,23H,6-7H2,1-2H3,(H,17,20)(H,18,24)(H,21,22)
Affinity DataIC50: 546nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair