BDBM93413 PHD Inhibitor, 8{3}

SMILES CC(C)C[C@@H](NC(C)=O)C(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1

InChI Key InChIKey=NGCNRBOGQFPBFY-OAHLLOKOSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 93413   

TargetEgl nine homolog 1(Homo sapiens (Human))
Amgen Inc

LigandPNGBDBM93413(PHD Inhibitor, 8{3})
Show SMILES CC(C)C[C@@H](NC(C)=O)C(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1
Show InChI InChI=1S/C22H28N4O7/c1-11(2)7-15(25-12(3)27)20(31)23-9-13-5-6-16-14(8-13)19(30)18(22(33)26(16)4)21(32)24-10-17(28)29/h5-6,8,11,15,30H,7,9-10H2,1-4H3,(H,23,31)(H,24,32)(H,25,27)(H,28,29)/t15-/m1/s1
Affinity DataIC50: 521nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair