BDBM93417 PHD Inhibitor, 8{7}

SMILES CC(=O)N[C@@H](CCCCN)C(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1

InChI Key InChIKey=IWJJDLNJDSEJFC-HNNXBMFYSA-N

Data  1 IC50

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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 93417   

TargetEgl nine homolog 1(Homo sapiens (Human))
Amgen Inc

LigandPNGBDBM93417(PHD Inhibitor, 8{7})
Show SMILES CC(=O)N[C@@H](CCCCN)C(=O)NCc1ccc2n(C)c(=O)c(C(=O)NCC(O)=O)c(O)c2c1
Show InChI InChI=1S/C22H29N5O7/c1-12(28)26-15(5-3-4-8-23)20(32)24-10-13-6-7-16-14(9-13)19(31)18(22(34)27(16)2)21(33)25-11-17(29)30/h6-7,9,15,31H,3-5,8,10-11,23H2,1-2H3,(H,24,32)(H,25,33)(H,26,28)(H,29,30)/t15-/m0/s1
Affinity DataIC50: 409nMAssay Description:PHD1,2,3 activity was measured utilizing homogeneous time-resolved fluroescence energy transfer techology by detecting the trans-4-hydroxylatio of HI...More data for this Ligand-Target Pair