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Found 199 Enz. Inhib. hit(s) with Target = 'Bifunctional protein GlmU'
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50294336(5-amino-2-(4-aminophenylamino)benzenesulfonic acid...)
Affinity DataKi:  17nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483325(CHEMBL1652297 | Mac0029665)
Affinity DataKi:  23nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50483326(CHEMBL1652296 | Mac0008028)
Affinity DataKi:  404nMAssay Description:Competitive inhibition of Acetyltransferase activity of Escherichia coli BL21(DE3) GlmU in presence of AcCoAMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  7nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075297(CHEMBL2207606)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075297(CHEMBL2207606)
Affinity DataIC50:  10nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92472(Sulfonamide, 3)
Affinity DataIC50:  18nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92472(Sulfonamide, 3)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92472(Sulfonamide, 3)
Affinity DataIC50:  20nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
TargetBifunctional protein GlmU(Haemophilus influenzae)
Astrazeneca

LigandPNGBDBM92474(Sulfonamide, 5)
Affinity DataIC50:  23nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50102673(CHEMBL3341771)
Affinity DataIC50:  27nMAssay Description:Inhibition of Escherichia coli ATCC 27325 GlmU expressed in Escherichia coli HMS174(DE3) incubated for 15 mins prior to MgCl2 addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075387(CHEMBL3415068)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075298(CHEMBL2207605)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075298(CHEMBL2207605)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075387(CHEMBL3415068)
Affinity DataIC50:  30nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075325(CHEMBL2207599)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075301(CHEMBL2207600)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075300(CHEMBL2207602)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075301(CHEMBL2207600)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075325(CHEMBL2207599)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075300(CHEMBL2207602)
Affinity DataIC50:  40nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075381(CHEMBL3415072)
Affinity DataIC50:  50nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075381(CHEMBL3415072)
Affinity DataIC50:  50nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM92473(Sulfonamide, 4)
Affinity DataIC50:  58nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075379(CHEMBL3415115)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075385(CHEMBL2207224)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075385(CHEMBL2207224)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075379(CHEMBL3415115)
Affinity DataIC50:  60nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075383(CHEMBL2207226)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075370(CHEMBL3414903)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075299(CHEMBL2207604)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075370(CHEMBL3414903)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075383(CHEMBL2207226)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075299(CHEMBL2207604)
Affinity DataIC50:  90nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075369(CHEMBL3414904)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075369(CHEMBL3414904)
Affinity DataIC50:  100nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50102677(CHEMBL3343057)
Affinity DataIC50:  120nMAssay Description:Inhibition of Escherichia coli ATCC 27325 GlmU expressed in Escherichia coli HMS174(DE3) incubated for 15 mins prior to MgCl2 addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075372(CHEMBL3414901)
Affinity DataIC50:  200nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075372(CHEMBL3414901)
Affinity DataIC50:  200nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50365095(CHEMBL1951184)
Affinity DataIC50:  250nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50365095(CHEMBL1951184)
Affinity DataIC50:  250nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50102714(CHEMBL3343050)
Affinity DataIC50:  260nMAssay Description:Inhibition of Escherichia coli ATCC 27325 GlmU expressed in Escherichia coli HMS174(DE3) incubated for 15 mins prior to MgCl2 addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Haemophilus influenzae)
Astrazeneca

LigandPNGBDBM92473(Sulfonamide, 4)
Affinity DataIC50:  280nMpH: 7.35Assay Description:Inhibition assay using GlmU bifuncation enzyme with various bacterial strains.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50102674(CHEMBL3343051)
Affinity DataIC50:  350nMAssay Description:Inhibition of Escherichia coli ATCC 27325 GlmU expressed in Escherichia coli HMS174(DE3) incubated for 15 mins prior to MgCl2 addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50102681(CHEMBL3343041)
Affinity DataIC50:  370nMAssay Description:Inhibition of Escherichia coli ATCC 27325 GlmU expressed in Escherichia coli HMS174(DE3) incubated for 15 mins prior to MgCl2 addition measured after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50075386(CHEMBL3415069)
Affinity DataIC50:  400nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50365098(CHEMBL1951187)
Affinity DataIC50:  400nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBifunctional protein GlmU(Escherichia coli)
Mcmaster University

Curated by ChEMBL
LigandPNGBDBM50365098(CHEMBL1951187)
Affinity DataIC50:  400nMAssay Description:Inhibition of Escherichia coli GlmU acetyltransferase activity assessed as coenzyme A production using acetyl CoA substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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