Compile Data Set for Download or QSAR
maximum 50k data
Found 35 Enz. Inhib. hit(s) with Target = 'Kinesin heavy chain isoform 5A'
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50252149((2S)-4-(2,5-difluorophenyl)-N-[(3R,4S)-3-fluoro-1-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of cloned human nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50383087(CHEMBL2031572)
Affinity DataIC50:  5.00E+4nMAssay Description:Inhibition of human Kif5A ATPase activity by pyruvate kinase/lactate dehydrogenase-linked assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293745(2-(4-sulfamoylphenylamino)-1-(1-(2-(trifluoromethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293746(1-(1-phenylcyclopropyl)-2-(4-sulfamoylphenylamino)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293747(1-(pyridin-2-ylmethyl)-2-(4-sulfamoylphenylamino)-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293748(1-(2-methoxybenzyl)-2-(4-sulfamoylphenylamino)-1H-...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293749(1-(2,3-dimethoxybenzyl)-2-(4-sulfamoylphenylamino)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293750(1-(benzo[d]thiazol-2-ylmethyl)-2-(4-sulfamoylpheny...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293751(1-((5-chlorobenzo[b]thiophen-3-yl)methyl)-2-(4-sul...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293752(1-(benzo[b]thiophen-3-ylmethyl)-2-(4-sulfamoylphen...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293753(2-(4-(methylsulfonyl)phenylamino)-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293754(2-(4-methoxyphenylamino)-1-(2-(trifluoromethyl)ben...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293755(2-(3-fluoro-4-methoxyphenylamino)-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293756(2-(4-(methylthio)phenylamino)-1-(2-(trifluoromethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293757(2-(4-sulfamoylphenylamino)-1-(2-(trifluoromethyl)b...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293758(2-(4-(methylsulfonyl)phenylamino)-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293759(2-(4-methoxyphenylamino)-1-(2-(trifluoromethyl)ben...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293760(2-(3-fluoro-4-methoxyphenylamino)-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293761(2-(4-(methylthio)phenylamino)-1-(2-(trifluoromethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293762(CHEMBL558477 | methyl 2-(4-sulfamoylphenylamino)-1...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293763(CHEMBL551230 | methyl 2-(4-methoxyphenylamino)-1-(...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293764(CHEMBL549531 | methyl 2-(4-(methylthio)phenylamino...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293765(2-(4-methoxyphenylamino)-N-methyl-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293766(CHEMBL562353 | N-methyl-2-(4-sulfamoylphenylamino)...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293767(CHEMBL559627 | N,N-dimethyl-2-(4-sulfamoylphenylam...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293768(4-(5-(pyrrolidine-1-carbonyl)-1-(2-(trifluoromethy...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293769(CHEMBL538431 | N-(2-methoxyphenyl)-2-(4-sulfamoylp...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293770(CHEMBL563993 | N-(2-methoxyphenyl)-2-(4-methoxyphe...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293771(2-(3-aminopyrrolidin-1-yl)-1-(2-(trifluoromethyl)b...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293772(2-(4-methylbenzylamino)-1-(2-(trifluoromethyl)benz...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293773(2-(4-methoxybenzylamino)-1-(2-(trifluoromethyl)ben...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293774(2-(4-(methylsulfonyl)benzylamino)-1-(2-(trifluorom...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293775(2-(4-sulfamoylbenzylamino)-1-(2-(trifluoromethyl)b...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293776(2-(2-morpholinoethylamino)-1-(2-(trifluoromethyl)b...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetKinesin heavy chain isoform 5A(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50293744(2-(4-sulfamoylphenylamino)-1-(2-(trifluoromethyl)b...)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of nKHCMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed