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Found 11 Enz. Inhib. hit(s) with Target = 'NADP-dependent malic enzyme'
TargetNADP-dependent malic enzyme(Escherichia coli (strain K12))
Institute Of Chemical Physics

Curated by ChEMBL
LigandPNGBDBM50338502(5-O-phosphate-1-N-(4'-(4''-methoxyhenyl))-[1',2',3...)
Affinity DataKi:  5.70E+4nMAssay Description:Inhibition of Escherichia coli K-12 recombinant NAD-dependent malic enzyme by Dixon plotMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177180(3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50:  150nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177175(1-benzyl-3-(4-(4-hydroxyphenyl)piperazin-1-yl)-1-p...)
Affinity DataIC50:  450nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177184(1-(3-chloro-4-methylphenyl)3-(4-(4-hydroxyphenyl)p...)
Affinity DataIC50:  560nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177177(1-phenyl-3-(4-(3-(trifluoromethyl)phenyl)piperazin...)
Affinity DataIC50:  3.15E+3nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177178(1-benzyl-3-(4-(3-hydroxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177179(3-(4-(4-fluorophenyl)piperazin-1-yl)-1-phenylpyrro...)
Affinity DataIC50:  1.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177182(1-benzyl-3-(4-(4-methoxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177176(1-benzyl-3-(4-(2-hydroxyphenyl)piperazin-1-yl)pyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177183(1-(2,3-dichlorophenyl)-3-(4-(4-methoxyphenyl)piper...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNADP-dependent malic enzyme(Homo sapiens (Human))
Cytrx Laboratories

Curated by ChEMBL
LigandPNGBDBM50177181(3-(4-(4-methoxyphenyl)piperazin-1-yl)-1-phenylpyrr...)
Affinity DataIC50: >2.00E+4nMAssay Description:Inhibitory activity against cytosolic malic enzymeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed