Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Neuropeptide Y-Y2 receptor'
TargetNeuropeptide Y-Y2 receptor(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50414468(CHEMBL1196581 | CHEMBL557502)
Affinity DataKi:  50.1nMAssay Description:Antagonist activity at rat NPY Y2 receptor expressed in HEK cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y-Y2 receptor(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417471(CHEMBL1287953)
Affinity DataKi:  63.1nMAssay Description:Antagonist activity at rat NPY Y2 receptor expressed in HEK cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuropeptide Y-Y2 receptor(Rattus norvegicus)
Glaxosmithkline

Curated by ChEMBL
LigandPNGBDBM50417475(CHEMBL1288016)
Affinity DataKi:  79.4nMAssay Description:Antagonist activity at rat NPY Y2 receptor expressed in HEK cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed