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Found 21 Enz. Inhib. hit(s) with Target = 'Quorum-sensing transcriptional repressor QscR'
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50373105(CHEMBL259441)
Affinity DataIC50:  30nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as inhibition of dodecanoyl homoserine lactone induced prod...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50373107(CHEMBL259439)
Affinity DataIC50:  130nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as inhibition of dodecanoyl homoserine lactone induced prod...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50373104(CHEMBL265683)
Affinity DataIC50:  160nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as inhibition of dodecanoyl homoserine lactone induced prod...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50373103(CHEMBL258913)
Affinity DataIC50:  180nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as inhibition of dodecanoyl homoserine lactone induced prod...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50373106(CHEMBL259440)
Affinity DataIC50:  200nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as inhibition of dodecanoyl homoserine lactone induced prod...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468432(CHEMBL4285396)
Affinity DataIC50: >2.50E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ tr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468426(CHEMBL3235593)
Affinity DataIC50: >2.50E+5nMAssay Description:Antagonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ tr...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468428(CHEBI:44612 | CHEMBL1234965)
Affinity DataEC50:  3.32E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sidPDB
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468425(CHEBI:56080 | CHEMBL208383)
Affinity DataEC50:  1.38E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoKEGGPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  15nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468429(CHEMBL4279608)
Affinity DataEC50:  815nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468431(CHEMBL408326)
Affinity DataEC50:  1.59E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50350703(CHEMBL1814828)
Affinity DataEC50:  80nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468427(CHEMBL1812101)
Affinity DataEC50:  359nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468424(CHEMBL4287516)
Affinity DataEC50:  3.46E+3nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351510(CHEMBL8463)
Affinity DataEC50:  78nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as production of beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351512(CHEMBL8483)
Affinity DataEC50:  22nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as production of beta-galactosidaseMore data for this Ligand-Target Pair
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351509(CHEMBL8799)
Affinity DataEC50:  6nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as production of beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351252(CHEMBL8755)
Affinity DataEC50:  5nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as production of beta-galactosidaseMore data for this Ligand-Target Pair
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50468430(CHEMBL4283085)
Affinity DataEC50:  834nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli JLD271 harboring QscR expression plasmid pJN105Q and pPA1897-lacZ trans...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetQuorum-sensing transcriptional repressor QscR(Pseudomonas aeruginosa)
University Of Wisconsin-Madison

Curated by ChEMBL
LigandPNGBDBM50351511(CHEMBL463321)
Affinity DataEC50:  11nMAssay Description:Agonist activity at Pseudomonas aeruginosa QscR expressed in Escherichia coli assessed as production of beta-galactosidaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed