TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 3.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 4.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 8nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 8.40nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 17.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 19.6nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 21.3nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 23.9nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 32.5nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataKi: 49.7nMAssay Description:Inhibition of PP1gamma by firefly bioluminescence assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataKi: >1.00E+3nM ΔG°: >-34.2kJ/molepH: 7.0 T: 2°CAssay Description:PTP activity was assayed using p-nitrophenyl phosphate (pNPP) as a substrate in DMG buffer (50 mM DMG, pH 7.0, 1 mM EDTA, 150 mM NaCl, 2 mM DTT, 0.1 ...More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-alpha catalytic subunit(Homo sapiens (Human))
3-Dimensional Pharmaceuticals
Curated by ChEMBL
3-Dimensional Pharmaceuticals
Curated by ChEMBL
Affinity DataKi: >6.70E+4nMAssay Description:In vitro inhibitory activity of the compound was tested against serine protease UrokinaseMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.30E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 4.30E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 4.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 5.70E+5nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.01E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.10E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.20E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.50E+6nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 1.70E+7nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase(Enterobacteria phage lambda)
Utah State University
Curated by ChEMBL
Utah State University
Curated by ChEMBL
Affinity DataKi: 2.00E+7nMAssay Description:Inhibitory activity against Serine/Threonine Protein Phosphatase (Lamda protein phosphatase)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.0100nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in E275RMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in wild typeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.0200nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D220VMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.0300nMAssay Description:Exogenous inhibition concentration of Serine/threonine protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B alpha isoform(Homo sapiens (Human))
University Of California
Curated by ChEMBL
University Of California
Curated by ChEMBL
Affinity DataIC50: 0.0650nMAssay Description:Observed inhibition activity of the compounds against protein phosphatases 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 56 kDa regulatory subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 0.0700nMAssay Description:Tested for inhibition of purified catalytic subunit of protein phosphatase-2A from human erythrocytesMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Exogenous inhibition concentration of Serine/threonine protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 56 kDa regulatory subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 0.100nMAssay Description:Tested for inhibition of purified catalytic subunit of protein phosphatase-2A from human erythrocytesMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 56 kDa regulatory subunit alpha isoform(Homo sapiens (Human))
TBA
Curated by ChEMBL
TBA
Curated by ChEMBL
Affinity DataIC50: 0.130nMAssay Description:Tested for inhibition of purified catalytic subunit of protein phosphatase-2A from human erythrocytesMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.140nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in D220VMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Observed inhibition activity against protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.200nMAssay Description:Exogenous inhibition concentration of Serine/threonine protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibition of microcystin analogues to catalytic subunits of Serine/threonine protein phosphatase 2A (PP2Ac)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A catalytic subunit alpha isoform(Bos taurus)
University Of California Irvine
Curated by ChEMBL
University Of California Irvine
Curated by ChEMBL
Affinity DataIC50: 0.300nMAssay Description:Inhibitory concentration of the compound against protein phosphatase 1 (PP1) using phosphorylase-a assayMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.400nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in E275RMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Observed inhibition activity against protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.450nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in wild typeMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.560nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in C127SMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 0.700nMAssay Description:Exogenous inhibition concentration of Serine/threonine protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase PP1-gamma catalytic subunit(Homo sapiens (Human))
Nagoya University
Curated by ChEMBL
Nagoya University
Curated by ChEMBL
Affinity DataIC50: 0.800nMAssay Description:Inhibition of Serine/threonine protein phosphatase 1 (PP1) mutants by natural toxins in Y272FMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition activity against protein phosphatase 2A (PP2A), activity taken from literatureMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Exogenous inhibition concentration of Serine/threonine protein phosphatase 2A (PP2A)More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Concentration required to inhibit the action of protein phosphatase 2AMore data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A activator(Homo sapiens (Human))
Indiana University Research And Technology
US Patent
Indiana University Research And Technology
US Patent
Affinity DataIC50: 1nMAssay Description:Protein phosphatase inhibitory activity of calyculin derivatives.More data for this Ligand-Target Pair
TargetSerine/threonine-protein phosphatase 2A 55 kDa regulatory subunit B(Gallus gallus)
The University Of Newcastle
Curated by ChEMBL
The University Of Newcastle
Curated by ChEMBL
Affinity DataIC50: 1nMAssay Description:Inhibition activity against protein phosphatase 2A (PP2A), activity taken from literatureMore data for this Ligand-Target Pair