Potent and highly selective neurokinin antagonists

MeSH terms

• Amino Acid Sequence
• Animals
• Guinea Pigs
• In Vitro Techniques
• Intestinal Mucosa / metabolism
• Intestines / drug effects
• Intestines / physiology
• Molecular Sequence Data
• Molecular Structure
• Muscle Contraction / drug effects
• Muscle, Smooth / drug effects
• Muscle, Smooth / metabolism
• Muscle, Smooth / physiology
• Neurokinin A / analogs & derivatives*
• Neurokinin A / antagonists & inhibitors*
• Neurokinin A / chemical synthesis
• Neurokinin A / pharmacology
• Neurokinin B / analogs & derivatives*
• Neurokinin B / antagonists & inhibitors*
• Neurokinin B / chemical synthesis
• Neurokinin B / pharmacology
• Protein Conformation
• Rats
• Receptors, Neurokinin-1
• Receptors, Neurokinin-2
• Receptors, Neurokinin-3
• Receptors, Neurotransmitter / drug effects
• Receptors, Neurotransmitter / metabolism
• Structure-Activity Relationship
• Substance P / analogs & derivatives*
• Substance P / antagonists & inhibitors*
• Substance P / chemical synthesis
• Substance P / pharmacology