Affinity DataIC50: 12nMAssay Description:Inhibition of recombinant human EGFR L858R mutant expressed in baculovirus infected insect cells preincubated for 5 mins followed by ATP addition and...More data for this Ligand-Target Pair
Affinity DataIC50: 13nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 23nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 27nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 34nMAssay Description:Inhibition of recombinant human EGFR L858R mutant expressed in baculovirus infected insect cells preincubated for 5 mins followed by ATP addition and...More data for this Ligand-Target Pair
Affinity DataIC50: 38nMAssay Description:Inhibition of recombinant human EGFR L858R mutant expressed in baculovirus infected insect cells preincubated for 5 mins followed by ATP addition and...More data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 46nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Al-Azhar University
Curated by ChEMBL
Al-Azhar University
Curated by ChEMBL
Affinity DataIC50: 91nMAssay Description:Inhibition of recombinant human GST-tagged HER2 (676-end) expressed in baculovirus infected Sf9 insect cells preincubated for 5 mins followed by ATP ...More data for this Ligand-Target Pair
Affinity DataIC50: 95nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 108nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 130nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human EGFR T790M mutant expressed in baculovirus infected Sf21 insect cells preincubated for 5 mins f...More data for this Ligand-Target Pair
Affinity DataIC50: 137nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human EGFR T790M mutant expressed in baculovirus infected Sf21 insect cells preincubated for 5 mins f...More data for this Ligand-Target Pair
Affinity DataIC50: 205nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 225nMAssay Description:Inhibition of N-terminal GST-tagged recombinant human EGFR T790M mutant expressed in baculovirus infected Sf21 insect cells preincubated for 5 mins f...More data for this Ligand-Target Pair
TargetReceptor tyrosine-protein kinase erbB-2(Homo sapiens (Human))
Al-Azhar University
Curated by ChEMBL
Al-Azhar University
Curated by ChEMBL
Affinity DataIC50: 240nMAssay Description:Inhibition of recombinant human GST-tagged HER2 (676-end) expressed in baculovirus infected Sf9 insect cells preincubated for 5 mins followed by ATP ...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1/2/3(Homo sapiens (Human))
Al-Azhar University
Curated by ChEMBL
Al-Azhar University
Curated by ChEMBL
Affinity DataIC50: 250nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR (789-end) expressed in baculovirus infected Sf9 insect cells preincubated for 5 mins followed by ATP...More data for this Ligand-Target Pair
TargetVascular endothelial growth factor receptor 1/2/3(Homo sapiens (Human))
Al-Azhar University
Curated by ChEMBL
Al-Azhar University
Curated by ChEMBL
Affinity DataIC50: 276nMAssay Description:Inhibition of GST-tagged recombinant human VEGFR (789-end) expressed in baculovirus infected Sf9 insect cells preincubated for 5 mins followed by ATP...More data for this Ligand-Target Pair
Affinity DataIC50: 358nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 493nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 751nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 993nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.18E+3nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 1.62E+3nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.89E+3nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.93E+3nMAssay Description:Inhibition of EGFR in human HepG2 cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8.26E+3nMAssay Description:Inhibition of EGFR (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 6.11E+4nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 8.60E+4nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 9.20E+4nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 1.03E+5nMAssay Description:Inhibition of EGFR L858R mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 3.77E+5nMAssay Description:Inhibition of EGFR T790M mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.21E+5nMAssay Description:Inhibition of EGFR T790M mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.33E+5nMAssay Description:Inhibition of EGFR T790M mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair
Affinity DataIC50: 4.62E+5nMAssay Description:Inhibition of EGFR T790M mutant (unknown origin) by FRET assayMore data for this Ligand-Target Pair