TargetSubstance-P receptor(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by PDSP Ki Database
Astrazeneca Pharmaceuticals
Curated by PDSP Ki Database
TargetSubstance-P receptor(Homo sapiens (Human))
Astrazeneca Pharmaceuticals
Curated by PDSP Ki Database
Astrazeneca Pharmaceuticals
Curated by PDSP Ki Database
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 200nMAssay Description:Inhibition of PDK1 (unknown origin) using PDKtide substrate and [gamma-32P]ATP by scintillation counting methodMore data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 600nMAssay Description:Inhibition of human platelet phosphodiesterase 3More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
Target3-phosphoinositide-dependent protein kinase 1(Homo sapiens (Human))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 4.90E+3nMAssay Description:Inhibition of PDK1 (unknown origin) expressed in HEK293 cells using PDKtide as substrate after 10 mins by liquid scintillation counting in presence o...More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 5.00E+3nMAssay Description:Inhibition of human platelet phosphodiesterase 2More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 6.00E+3nMAssay Description:Inhibition of human platelet phosphodiesterase 2More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 9.00E+3nMAssay Description:Inhibition of human platelet phosphodiesterase 2More data for this Ligand-Target Pair
TargetcGMP-dependent 3',5'-cyclic phosphodiesterase(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 4.00E+4nMAssay Description:Inhibition of human platelet phosphodiesterase 2More data for this Ligand-Target Pair
TargetcGMP-inhibited 3',5'-cyclic phosphodiesterase 3A/3B(Homo sapiens (Human))
Monash University
Curated by ChEMBL
Monash University
Curated by ChEMBL
Affinity DataIC50: 1.00E+5nMAssay Description:Inhibition of human platelet phosphodiesterase 3More data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataIC50: 1.40E+5nMAssay Description:Inhibition of Escherichia coli DsbA using DOTA/Eu(III)-CQQGFDGTQNSCK-MCA as substrate in presence of oxidized glutathione measured by fluorescence an...More data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: >1.00E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 4.60E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 4.03E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 5.31E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 2.74E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 9.78E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 8.20E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 2.30E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 1.10E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 8.30E+5nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair
TargetThiol:disulfide interchange protein DsbA(Escherichia coli (strain K12))
La Trobe University
Curated by ChEMBL
La Trobe University
Curated by ChEMBL
Affinity DataKd: 1.14E+6nMAssay Description:Binding affinity to 15N-labelled Escherichia coli DsbA measured by 1H-15N HSQC NMR spectroscopyMore data for this Ligand-Target Pair