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Found 7 with Last Name = 'acosta' and Initial = 'lm'
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50041978(CHEMBL3134157)
Affinity DataKi:  3.60nMAssay Description:Inhibition of human C-terminal His6-tagged SphK1 expressed in baculovirus infected Sf21 insect cellsMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50443389(CHEMBL2376441)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of V5-His-tagged human SphK1 using sphingosine as substrate in presence of [gamma-32P]ATPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50312869(4-(4-(4-chlorophenyl)thiazol-2-ylamino)phenol | CH...)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibition of recombinant human GST-tagged SphK1 using [3H]-sphingosine as substrate after 30 mins by scintillation counting methodMore data for this Ligand-Target Pair
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50443387(CHEMBL3086811)
Affinity DataIC50:  3.60E+3nMAssay Description:Inhibition of SphK1 (unknown origin) expressed in HEK293 cells using sphingosine as substrate after 30 mins in presence of [gamma-32P]ATP by Cerenkov...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50277232(CHEMBL4170798)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of human N-terminal MGHHHHHHHHHHSSG-tagged SphK1 (2 to 384 residues) expressed in Escherichia coli Rosetta-2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50277231(CHEMBL4162455)
Affinity DataIC50:  5.50E+4nMAssay Description:Inhibition of human N-terminal MGHHHHHHHHHHSSG-tagged SphK1 (2 to 384 residues) expressed in Escherichia coli Rosetta-2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSphingosine kinase 1(Homo sapiens (Human))
Universidad Nacional De San Luis

Curated by ChEMBL
LigandPNGBDBM50277230(CHEMBL4173139)
Affinity DataIC50:  6.00E+4nMAssay Description:Inhibition of human N-terminal MGHHHHHHHHHHSSG-tagged SphK1 (2 to 384 residues) expressed in Escherichia coli Rosetta-2 by fluorescence assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed