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Found 19 with Last Name = 'adanitsch' and Initial = 'f'
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326399((+/-)-trans-4-Butyl-1-[(9-deazaadenin-9-yl)methyl]...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326399((+/-)-trans-4-Butyl-1-[(9-deazaadenin-9-yl)methyl]...)
Affinity DataKi:  0.800nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326400((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-3-hydro...)
Affinity DataKi:  1.70nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326402((+/-)-trans-4-Cyclopropyl-1-[(9-deazaadenin-9-yl)m...)
Affinity DataKi:  2.10nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326403((+/-)-trans-4-Cyclopentyl-1-[(9-deazaadenin-9-yl)m...)
Affinity DataKi:  2.60nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326407((+/-)-trans-4-Allyl-1-[(9-deazaadenin-9-yl)methyl]...)
Affinity DataKi:  3nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326398((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-4-ethyl...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326398((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-4-ethyl...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326406((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-3-hydro...)
Affinity DataKi:  3.20nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326405((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-3-hydro...)
Affinity DataKi:  8nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326404((+/-)-trans-4-(Cyclohexylmethyl)-1-[(9-deaza-adeni...)
Affinity DataKi:  14nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326401((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-3-hydro...)
Affinity DataKi:  18nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326408((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-4-ethyn...)
Affinity DataKi:  31nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326411((+/-)-Benzyl cis-3-(Benzoyloxy)-4-ethylpyrrolidine...)
Affinity DataKi:  34nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326409((+/-)-trans-1-[(9-Deazaadenin-9-yl)methyl]-3-hydro...)
Affinity DataKi:  59nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetS-methyl-5'-thioadenosine phosphorylase(Homo sapiens (Human))
Industrial Research

Curated by ChEMBL
LigandPNGBDBM50326410((+/-)-trans-4-[3-(Benzylthio)propyl]-1-[(9-deazaad...)
Affinity DataKi:  71nMAssay Description:Inhibition of His-tagged human MTAPMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of Natural Resources And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50028262(CHEMBL3354640)
Affinity DataEC50:  0.0800nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 cells coexpressed with human MD2/CD14 assessed as activation of NFkappaB signaling after 20 to 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of Natural Resources And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50028261(CHEMBL3354639)
Affinity DataEC50:  0.400nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 cells coexpressed with human MD2/CD14 assessed as activation of NFkappaB signaling after 20 to 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetToll-like receptor 4(Homo sapiens (Human))
University Of Natural Resources And Life Sciences

Curated by ChEMBL
LigandPNGBDBM50028263(CHEMBL3354641)
Affinity DataEC50:  31nMAssay Description:Agonist activity at human TLR4 expressed in HEK293 cells coexpressed with human MD2/CD14 assessed as activation of NFkappaB signaling after 20 to 24 ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed