TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: 9.5nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: 26.9nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: 48nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: 52nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: 180nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University
Curated by ChEMBL
Philipps University
Curated by ChEMBL
Affinity DataIC50: >500nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair