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Found 6 with Last Name = 'adhikary' and Initial = 't'
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  9.5nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383371(CHEMBL2030550)
Affinity DataIC50:  26.9nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383373(CHEMBL592652 | GSK0660)
Affinity DataIC50:  48nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  52nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383370(CHEMBL2030543)
Affinity DataIC50:  180nMAssay Description:Displacement of fluormone Pan-PPAR Green from mouse recombinant GST-tagged PPARbeta/delta LBD after 60 mins by TR-FRET assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Mus musculus)
Philipps University

Curated by ChEMBL
LigandPNGBDBM50383372(CHEMBL1998001)
Affinity DataIC50: >500nMAssay Description:Inverse agonist activity at PPARbeta/delta in mouse C2C12 cells assessed as inhibition of Angptl4 expression after 24 hrs by RT-qPCR analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed