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Found 166 with Last Name = 'adolfs' and Initial = 'tj'
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM50004108((+-)-nicotine | (R,S)-nicotine | (RS)-nicotine | 3...)
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50230537((S)-3-(4-chlorophenyl)-N'-(4-chlorophenylsulfonyl)...)
Affinity DataKi:  7.80nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86831((+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  10nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86826((S)-5-(5-methoxypyridin-3-yl)-N-methylpent-4-en-2-...)
Affinity DataKi:  11nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138899(3-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  13.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163112(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-ethy...)
Affinity DataKi:  14nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86831((+/-)-2-(pyrrolidin-3-yl)-1H-pyrrolo[2,3-b]pyridin...)
Affinity DataKi:  16nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138902(CHEMBL160767 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  16.1nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138903(CHEMBL350924 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  16.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163139(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  19nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138897(CHEMBL351123 | Naphthalene-2-sulfonic acid 1-[3-(4...)
Affinity DataKi:  21.8nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138921(CHEMBL158138 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  22.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163132(5-Bromo-1-(4-chloro-phenyl)-2-(2,4-dichloro-phenyl...)
Affinity DataKi:  23nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50140220(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-1H-imi...)
Affinity DataKi:  23nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172907(3,4-diarylpyrazoline derivative | CHEMBL383580)
Affinity DataKi:  24nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138912(CHEMBL156556 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  24.2nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM29094((+/-)-SLV319 | (S)-3-(4-chlorophenyl)-N-(4-chlorop...)
Affinity DataKi:  25nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM21278(5-(4-chlorophenyl)-1-(2,4-dichlorophenyl)-4-methyl...)
Affinity DataKi:  25nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMedDrugBank

TargetNeuronal acetylcholine receptor subunit alpha-4(Rattus norvegicus (Rat))
Solvay Pharmaceuticals

Curated by PDSP Ki Database
LigandPNGBDBM86833(CAS_5310967 | Methyl-((E)-4-pyridin-3-yl-but-3-eny...)
Affinity DataKi:  26nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163119(5-Chloro-1-(4-chloro-phenyl)-2-(2,4-dichloro-pheny...)
Affinity DataKi:  27nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163111(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  27nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163140(2-(2,4-Dichloro-phenyl)-5-methyl-1-(4-trifluoromet...)
Affinity DataKi:  29nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163122(1-(4-Chloro-phenyl)-5-cyano-2-(2,4-dichloro-phenyl...)
Affinity DataKi:  30nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172899(3,4-diarylpyrazoline derivative | CHEMBL195050)
Affinity DataKi:  30nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163120(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  30nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172906(3,4-diarylpyrazoline derivative | CHEMBL371829)
Affinity DataKi:  32nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163138(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  33nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163117(CHEMBL175291 | [1-(4-Chloro-phenyl)-2-(2,4-dichlor...)
Affinity DataKi:  34nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163115(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  35nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163126(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  35nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138915(CHEMBL156264 | N-[1-[(S)-3-(4-Chloro-phenyl)-4-phe...)
Affinity DataKi:  35.9nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163136(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-fluo...)
Affinity DataKi:  36nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138900(CHEMBL157591 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  36.5nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50140232(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  40nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163128(2-(2,4-Dichloro-phenyl)-1-(4-fluoro-phenyl)-5-meth...)
Affinity DataKi:  52nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138919(CHEMBL158502 | N-[1-Amino-1-[3-(4-chloro-phenyl)-4...)
Affinity DataKi:  52.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163139(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  54nMAssay Description:In vitro displacement of CP-55940 binding to human CB2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138918(CHEMBL348174 | N-[1-[3-(4-Chloro-phenyl)-4-phenyl-...)
Affinity DataKi:  54.2nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163134(1-(5-Chloro-pyridin-2-yl)-2-(2,4-dichloro-phenyl)-...)
Affinity DataKi:  55nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50312823((S)-3-(4-chlorophenyl)-N-methyl-4-phenyl-N'-(piper...)
Affinity DataKi:  58nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163129(1-(4-Bromo-phenyl)-2-(2,4-dichloro-phenyl)-5-methy...)
Affinity DataKi:  60nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172897(3,4-diarylpyrazoline derivative | CHEMBL194566)
Affinity DataKi:  60nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163124(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  64nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138923(4-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  70.6nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50172910(3,4-diarylpyrazoline derivative | CHEMBL194351)
Affinity DataKi:  75nMAssay Description:Displacement of specific CP-55940 binding in CHO cells stably transfected with human cannabinoid receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50138909(2-Chloro-N-[1-[3-(4-chloro-phenyl)-4-phenyl-4,5-di...)
Affinity DataKi:  75.4nMAssay Description:Displacement of CP-55,940 binding from recombinant human cannabinoid receptor 1 expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163135(1-(4-Chloro-phenyl)-2-(2,4-dichloro-phenyl)-5-meth...)
Affinity DataKi:  94nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Solvay Pharma

Curated by ChEMBL
LigandPNGBDBM50163133(2-(2,4-Dichloro-phenyl)-1-(4-methoxy-phenyl)-5-met...)
Affinity DataKi:  106nMAssay Description:In vitro displacement of CP-55940 binding to human CB1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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