TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 10nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 50nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 80nMAssay Description:Inhibition of P-gp in human CMEC/D3 cells using calcein-AM as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 90nMAssay Description:Inhibition of P-gp in human CMEC/D3 cells using NBD-Aba as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 300nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 360nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 370nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 400nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 410nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 410nMAssay Description:Inhibition of P-gp in human CMEC/D3 cells using NBD-Aba as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 500nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 500nMAssay Description:Inhibition of P-gp in human 12D7-MDR cells using calcein-AM as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 510nMAssay Description:Inhibition of P-gp in human 12D7-MDR cells using NBD-Aba as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 520nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 570nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 590nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 590nMAssay Description:Inhibition of P-gp in human CMEC/D3 cells using calcein-AM as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 630nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 640nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 650nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 650nMAssay Description:Inhibition of P-gp in human 12D7-MDR cells using NBD-Aba as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 680nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 690nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 720nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 740nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 750nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 770nMAssay Description:Inhibition of P-gp in human 12D7-MDR cells using calcein-AM as substrate after 30 mins by flow cytometric analysisMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 770nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 820nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 870nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.02E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.04E+3nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.09E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.12E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.16E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
Affinity DataIC50: 1.20E+3nMAssay Description:Inhibition of P-gp in human 12D7-MDR cells using calcein-AM as substrateMore data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.23E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.24E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.26E+3nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.28E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.34E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Homo sapiens (Human))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.38E+3nMAssay Description:Inhibition of human erythrocyte AChE using ATCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.43E+3nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair
TargetCholinesterase(Equus caballus (Horse))
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
The Maharaja Sayajirao University Of Baroda
Curated by ChEMBL
Affinity DataIC50: 1.50E+3nMAssay Description:Inhibition of equine serum BuChE using BTCI as substrate preincubated for 30 mins followed by substrate addition measured after 30 mins by Ellman ass...More data for this Ligand-Target Pair