Affinity DataKi: 2.60E+4nMAssay Description:Displacement of [3H]QNB from M1 receptor in Wistar rat cerebral cortex homogenateMore data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 110nMAssay Description:Antagonist activity at CCR4More data for this Ligand-Target Pair
TargetC-C chemokine receptor type 4(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 140nMAssay Description:Antagonist activity at CCR4More data for this Ligand-Target Pair
TargetTyrosine-protein phosphatase non-receptor type 1(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 480nMAssay Description:Inhibition of GST-tagged PTP1B using pNPP as substrate by spectrophotometric analysisMore data for this Ligand-Target Pair
TargetTYR_PHOSPHATASE_2 domain-containing protein(Mycobacterium tuberculosis)
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataIC50: 1.10E+3nMAssay Description:Inhibition of Mycobacterium tuberculosis protein tyrosine phosphatase BMore data for this Ligand-Target Pair
Affinity DataIC50: 1.43E+5nMAssay Description:Displacement of [3H]QNB from M1 receptor in Wistar rat cerebral cortex homogenateMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataEC50: 80nMAssay Description:Agonist activity at human FSH receptor by cAMP-based assayMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataEC50: 50nMAssay Description:Agonist activity at human FSH receptor by aromatase-based assayMore data for this Ligand-Target Pair
TargetFollicle-stimulating hormone receptor(Homo sapiens (Human))
Dr. Hari Singh Gour University
Curated by ChEMBL
Dr. Hari Singh Gour University
Curated by ChEMBL
Affinity DataEC50: 1nMAssay Description:Allosteric activation of human FSH receptorMore data for this Ligand-Target Pair