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Found 301 with Last Name = 'ahmed' and Initial = 'e'
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Minia University

Curated by ChEMBL
LigandPNGBDBM50005480((-)-combretastatin | (Z)-3'-hydroxy-3,4,4',5-tetra...)
Affinity DataKi:  140nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Minia University

Curated by ChEMBL
LigandPNGBDBM50504214(CHEMBL4530425)
Affinity DataKi:  150nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSimilar to alpha-tubulin isoform 1(Bos taurus)
Minia University

Curated by ChEMBL
LigandPNGBDBM50504215(CHEMBL4463939)
Affinity DataKi:  260nMAssay Description:Inhibition of [3H] colchicine binding to bovine brain tubulin incubated for 30 mins by scintillation proximity assayMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  440nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176468(CHEMBL202223 | haloxysterol B)
Affinity DataKi:  850nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176465(CHEMBL382961 | haloxysterol C)
Affinity DataKi:  1.10E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176467(CHEMBL201253 | haloxysterol D)
Affinity DataKi:  2.20E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176468(CHEMBL202223 | haloxysterol B)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176470(24-ethyl-cholest-7-ene-3,5,6-triol | CHEMBL201951)
Affinity DataKi:  2.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176472(CHEMBL202496 | lawsaritol)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176466(24-ethylcholest-6-ene-3,5-diol | CHEMBL201866)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176466(24-ethylcholest-6-ene-3,5-diol | CHEMBL201866)
Affinity DataKi:  4.20E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176469(CHEMBL202221 | haloxysterol A)
Affinity DataKi:  4.50E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176473((24S)-ethylcholesta-7,9(11),22(E)-triene-3b-ol | C...)
Affinity DataKi:  4.60E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176471(5alpha,8alpha-epidioxy-(24S)-ethylcholesta-6,9(11)...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176469(CHEMBL202221 | haloxysterol A)
Affinity DataKi:  7.60E+3nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM10404((1S,12S,14R)-9-methoxy-4-methyl-11-oxa-4-azatetrac...)
Affinity DataKi:  8.00E+3nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176470(24-ethyl-cholest-7-ene-3,5,6-triol | CHEMBL201951)
Affinity DataKi:  1.26E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176472(CHEMBL202496 | lawsaritol)
Affinity DataKi:  1.61E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176467(CHEMBL201253 | haloxysterol D)
Affinity DataKi:  1.70E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCarboxylic ester hydrolase(Equus caballus (Horse))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176465(CHEMBL382961 | haloxysterol C)
Affinity DataKi:  1.80E+4nMAssay Description:Inhibitory activity against BuChE from horse serumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176473((24S)-ethylcholesta-7,9(11),22(E)-triene-3b-ol | C...)
Affinity DataKi:  2.06E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Karachi

Curated by ChEMBL
LigandPNGBDBM50176471(5alpha,8alpha-epidioxy-(24S)-ethylcholesta-6,9(11)...)
Affinity DataKi:  2.55E+4nMAssay Description:Inhibitory activity against AChE from electric eelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016564(CHEMBL3272448)
Affinity DataKi:  3.16E+4nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine N-methyltransferase(Cavia porcellus)
TBA

Curated by ChEMBL
LigandPNGBDBM50016547(CHEMBL3272447)
Affinity DataKi:  2.47E+5nMAssay Description:Inhibition of histamine N-methyltransferase in guinea pig brain using S-adenosyl-L-methionine-14C as substrate by scintillation spectrophotometerMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073539(CHEMBL3408926)
Affinity DataIC50:  1.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073512(CHEMBL3408911)
Affinity DataIC50:  1.70nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073531(CHEMBL3408918)
Affinity DataIC50:  2.90nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073533(CHEMBL3408920)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM15581(CHEMBL8706 | CLG | CLORGILINE | Clorgyline | N-[3-...)
Affinity DataIC50:  3.10nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073532(CHEMBL3408919)
Affinity DataIC50:  3.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073534(CHEMBL3408921)
Affinity DataIC50:  3.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073535(CHEMBL3408922)
Affinity DataIC50:  6.60nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073540(CHEMBL3408927)
Affinity DataIC50:  7.30nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073536(CHEMBL3408923)
Affinity DataIC50:  8.40nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM5445(CHEMBL554 | GW572016 | LAPATINIB DITOSYLATE | Lapa...)
Affinity DataIC50:  15nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50512093(CHEMBL4442101)
Affinity DataIC50:  16nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM11639(4-[5-(4-methylphenyl)-3-(trifluoromethyl)-1H-pyraz...)
Affinity DataIC50:  18nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50512095(CHEMBL4435643)
Affinity DataIC50:  18nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50512097(CHEMBL4536976)
Affinity DataIC50:  19nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50512102(CHEMBL4465207)
Affinity DataIC50:  20nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetPlatelet-derived growth factor receptor beta(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM50566726(CHEMBL4868909)
Affinity DataIC50:  20nMAssay Description:Inhibition of PDGFRbeta (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1/2/3/4(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM50566726(CHEMBL4868909)
Affinity DataIC50:  21nMAssay Description:Inhibition of FGFR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073537(CHEMBL3408924)
Affinity DataIC50:  22nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetFibroblast growth factor receptor 1/2/3/4(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM2579((2S,3R,4R,6R)-3-methoxy-2-methyl-4-(methylamino)-2...)
Affinity DataIC50:  27nMAssay Description:Inhibition of FGFR (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetEpidermal growth factor receptor(Homo sapiens (Human))
Egyptian National Research Centre

Curated by ChEMBL
LigandPNGBDBM50566726(CHEMBL4868909)
Affinity DataIC50:  33nMAssay Description:Inhibition of EGFR (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073510(CHEMBL3408909)
Affinity DataIC50:  34nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAmine oxidase [flavin-containing] A(Bos taurus)
Alexandria University

Curated by ChEMBL
LigandPNGBDBM50073543(CHEMBL3408930)
Affinity DataIC50:  36nMAssay Description:Inhibition of bovine brain MAO-A preincubated for 60 mins before substrate addition by fluorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Homo sapiens (Human))
Cairo University

Curated by ChEMBL
LigandPNGBDBM50512098(CHEMBL4574755)
Affinity DataIC50:  37nMAssay Description:Inhibition of human COX2 assessed as reduction in PGF2alpha production using arachidonic acid as substrate preincubated with enzyme for 10 mins follo...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMitogen-activated protein kinase 11/12/13/14(Homo sapiens (Human))
National Research Centre

Curated by ChEMBL
LigandPNGBDBM50537171(CHEMBL4576947)
Affinity DataIC50:  40nMAssay Description:Inhibition of p38alpha MAPK (unknown origin) using ATF-2 as substrate after 1 hr by ELISAMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
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