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Found 58 with Last Name = 'akaho' and Initial = 'e'
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  30nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85624(Indole ester derivative, 4 | Indole ester derivati...)
Affinity DataIC50:  1.34E+3nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197708(4-amino-N-(4-chlorophenyl)-N-methylbenzenesulfonam...)
Affinity DataIC50:  3.20E+3nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM17638(2-{1-[(4-chlorophenyl)carbonyl]-5-methoxy-2-methyl...)
Affinity DataIC50:  7.70E+3nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197704(CHEMBL227544 | N-(4-aminophenyl)-4-chloro-N-methyl...)
Affinity DataIC50:  9.20E+3nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197705(4-amino-N-(4-chlorophenyl)benzenesulfonamide | CHE...)
Affinity DataIC50:  1.20E+4nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479240(CHEMBL387906)
Affinity DataIC50:  1.21E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479247(CHEMBL225616)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197707(CHEMBL389184 | N-(4-amino-2-methoxyphenyl)-4-chlor...)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85644(Indole ester derivative, 24)
Affinity DataIC50:  2.14E+4nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197706(CHEMBL227545 | N-(4-amino-2-methylphenyl)-4-chloro...)
Affinity DataIC50:  2.60E+4nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479236(CHEMBL510682)
Affinity DataIC50:  3.91E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479239(CHEMBL225561)
Affinity DataIC50:  4.31E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479237(CHEMBL228722)
Affinity DataIC50:  6.63E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479234(CHEMBL503817)
Affinity DataIC50:  8.19E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479235(CHEMBL511479)
Affinity DataIC50:  8.47E+4nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197706(CHEMBL227545 | N-(4-amino-2-methylphenyl)-4-chloro...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoate | 2-(acetyloxy)benzoic acid ...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197708(4-amino-N-(4-chlorophenyl)-N-methylbenzenesulfonam...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197705(4-amino-N-(4-chlorophenyl)benzenesulfonamide | CHE...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197704(CHEMBL227544 | N-(4-aminophenyl)-4-chloro-N-methyl...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 2(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM50197707(CHEMBL389184 | N-(4-amino-2-methoxyphenyl)-4-chlor...)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of ovine COX2More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProstaglandin G/H synthase 1(Ovis aries (Sheep))
Okayama University Graduate School Of Medicine

Curated by ChEMBL
LigandPNGBDBM22360(2-(acetyloxy)benzoate | 2-(acetyloxy)benzoic acid ...)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of ovine COX1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50366348(CHEMBL1233654)
Affinity DataIC50:  1.30E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479244(CHEMBL509048)
Affinity DataIC50:  1.67E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479248(CHEMBL505693)
Affinity DataIC50:  1.70E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479242(CHEMBL472210)
Affinity DataIC50:  1.84E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479241(CHEMBL471503)
Affinity DataIC50:  1.97E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85623(Indole ester derivative, 3 | Indole ester derivati...)
Affinity DataIC50:  2.15E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479246(CHEMBL471341)
Affinity DataIC50: >2.40E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85633(Indole ester derivative, 13 | Indole ester derivat...)
Affinity DataIC50:  2.58E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479245(CHEMBL471512)
Affinity DataIC50: >2.73E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85634(Indole ester derivative, 14 | Indole ester derivat...)
Affinity DataIC50:  2.79E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85634(Indole ester derivative, 14 | Indole ester derivat...)
Affinity DataIC50:  3.06E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479243(CHEMBL471502)
Affinity DataIC50: >3.29E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50479238(CHEMBL504942)
Affinity DataIC50:  3.34E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProtein kinase C zeta type(Rattus norvegicus)
Okayama University

Curated by ChEMBL
LigandPNGBDBM50438882(10-Phenylpyrimido[4,5-b]quinoline-2,4(3H,10H)-dion...)
Affinity DataIC50: >3.45E+5nMAssay Description:Inhibition of rat brain protein kinase CMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85645(Indole ester derivative, 25 | Indole ester derivat...)
Affinity DataIC50: >5.00E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85646(Indole ester derivative, 26)
Affinity DataIC50: >5.00E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85621(Indole ester derivative, 1 | Indole ester derivati...)
Affinity DataIC50: >5.00E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85624(Indole ester derivative, 4 | Indole ester derivati...)
Affinity DataIC50:  5.13E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85622(Indole ester derivative, 2 | Indole ester derivati...)
Affinity DataIC50:  6.14E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85621(Indole ester derivative, 1 | Indole ester derivati...)
Affinity DataIC50:  6.31E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85632(Indole ester derivative, 12 | Indole ester derivat...)
Affinity DataIC50:  8.17E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85645(Indole ester derivative, 25 | Indole ester derivat...)
Affinity DataIC50:  8.30E+5nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85632(Indole ester derivative, 12 | Indole ester derivat...)
Affinity DataIC50: >1.00E+6nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85622(Indole ester derivative, 2 | Indole ester derivati...)
Affinity DataIC50: >1.00E+6nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85631(Indole ester derivative, 11 | Indole ester derivat...)
Affinity DataIC50: >1.00E+6nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85634(Indole ester derivative, 14 | Indole ester derivat...)
Affinity DataIC50: >1.00E+6nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Gallus gallus (Chicken))
Kobe Gakuin University

LigandPNGBDBM85631(Indole ester derivative, 11 | Indole ester derivat...)
Affinity DataIC50: >1.00E+6nMT: 2°CAssay Description:Takara Universal Tyrosine Assay Kit (Takara-bio co) was used to test the synthesized compounds. This assay kit determines the inhibition activities ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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