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Found 50 with Last Name = 'akhtar' and Initial = 'ms'
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50065646(CHEMBL3087181)
Affinity DataIC50: <0.400nMAssay Description:Inhibition of human MAGLMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50242634(5-((biphenyl-4-yl)methyl)-N,N-dimethyl-2H-tetrazol...)
Affinity DataIC50:  0.900nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM179929(US9133148, 1a)
Affinity DataIC50:  5.90nMAssay Description:Inhibition of human MAGL transfected in human HEK293T cells assessed as reduction in ABPP binding by competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM60622(BDBM50300355 | US11753371, Compound JZL-184 | US91...)
Affinity DataIC50:  6nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563791(CHEMBL4778803)
Affinity DataIC50:  6.5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563792(CHEMBL4788586)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563794(CHEMBL4793668)
Affinity DataIC50:  8nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563790(CHEMBL4780294)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563793(CHEMBL4793997)
Affinity DataIC50:  9nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563801(CHEMBL4779678)
Affinity DataIC50:  16nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563802(CHEMBL4793265)
Affinity DataIC50:  17nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  20nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563803(CHEMBL4797565)
Affinity DataIC50:  22nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563795(CHEMBL4786239)
Affinity DataIC50:  68nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563785(CHEMBL4792393)
Affinity DataIC50:  74nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50432829(CHEMBL2171700)
Affinity DataIC50:  78nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563809(CHEMBL4794817)
Affinity DataIC50:  117nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563797(CHEMBL4777523)
Affinity DataIC50:  151nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563808(CHEMBL4793077)
Affinity DataIC50:  196nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563796(CHEMBL4780477)
Affinity DataIC50:  242nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563800(CHEMBL4776276)
Affinity DataIC50:  282nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50414921(CHEMBL570812)
Affinity DataIC50:  424nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563799(CHEMBL4785038)
Affinity DataIC50:  780nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563798(CHEMBL4800406)
Affinity DataIC50:  815nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563788(CHEMBL4798413)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563787(CHEMBL4788417)
Affinity DataIC50:  6.50E+3nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563786(CHEMBL4783652)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563782(CHEMBL4786879)
Affinity DataIC50:  2.40E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50128581(Biphenyl-3-yl-carbamic acid cyclohexyl ester | CHE...)
Affinity DataIC50:  2.80E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50274981(4-(4,5-dihydrothiazol-2-yl)phenyl butylcarbamate |...)
Affinity DataIC50:  3.10E+4nMAssay Description:Inhibition of MAGL (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563781(CHEMBL4800077)
Affinity DataIC50:  3.70E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470016(CHEMBL288505)
Affinity DataIC50:  3.90E+4nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50101816(CHEBI:8107 | Dilabid | Dilantin | Dilantin-125 | D...)
Affinity DataIC50:  4.00E+4nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563784(CHEMBL4796478)
Affinity DataIC50:  4.70E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563783(CHEMBL4777889)
Affinity DataIC50:  4.80E+4nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563789(CHEMBL4799435)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563807(CHEMBL4777402)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563806(CHEMBL4783153)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563805(CHEMBL4784727)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetMonoglyceride lipase(Homo sapiens (Human))
Hamdard University

Curated by ChEMBL
LigandPNGBDBM50563804(CHEMBL4800531)
Affinity DataIC50: >1.00E+5nMAssay Description:Inhibition of human MAGL using 4-Nitrophenylacetate as substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470014(CHEMBL39010)
Affinity DataIC50:  1.03E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50003659(5H-dibenzo[b,f]azepine-5-carboxamide | CARBAMAZEPI...)
Affinity DataIC50:  1.31E+5nMAssay Description:Displacement of [3H]batrachotoxin A 20alpha-benzoate (BTX-B) from rat cerebral cortex voltage-gated sodium channelMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470017(CHEMBL1169567)
Affinity DataIC50:  1.60E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470011(CHEMBL288861)
Affinity DataIC50:  1.62E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470013(CHEMBL39810)
Affinity DataIC50:  2.85E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50227240(CHEMBL70727)
Affinity DataIC50:  3.80E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470015(CHEMBL39126)
Affinity DataIC50:  4.27E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50227231(CHEMBL41666)
Affinity DataIC50:  5.00E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50470012(CHEMBL38675)
Affinity DataIC50:  7.00E+5nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSodium channel protein type 1/2/3 subunit alpha(Rattus norvegicus)
University Of Alabama At Birmingham

Curated by ChEMBL
LigandPNGBDBM50227239(Tridione | Trimethadione | Troxidone)
Affinity DataIC50: >1.00E+6nMAssay Description:Inhibition of binding to sodium channel of rat cerebral cortexMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed