Affinity DataKi: 1nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.60nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 1.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.40nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 2.60nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 2.90nMAssay Description:Binding affinity to rat 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.20nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 4.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 5.10nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 5.70nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.30nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.5nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 6.80nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 7.70nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 8.20nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 8.70nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 10nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 10.1nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 10.8nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 12nMAssay Description:Binding affinity towards Alpha-1 adrenergic receptor in rat brain using [3H]prazosinMore data for this Ligand-Target Pair
Affinity DataKi: 12.4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 13.2nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15.3nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 15.9nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT7 receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 17.6nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 18.3nMAssay Description:Binding affinity to histamine H1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 19nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Binding affinity towards human recombinant adenosine A2A receptor by displacement of [3H]-SCH-58,261 radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 22.2nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22.2nMAssay Description:Binding affinity to human 5HT5A receptorMore data for this Ligand-Target Pair
Affinity DataKi: 22.9nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 23.3nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 24nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Homo sapiens (Human))
F. Hoffmann-La Roche
Curated by ChEMBL
F. Hoffmann-La Roche
Curated by ChEMBL
Affinity DataKi: 24nMAssay Description:In vitro binding affinity towards Alpha-1 adrenergic receptor by displacing [3H]prazosin radioligandMore data for this Ligand-Target Pair
Affinity DataKi: 24.8nMAssay Description:Binding affinity to human 5HT7 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 25.4nMAssay Description:Displacement of [3H]LSD from human recombinant 5HT5A receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair
Affinity DataKi: 26nMAssay Description:Displacement of [3H]mesulergine from human recombinant 5HT2C receptor expressed in HEK293-EBNA cellsMore data for this Ligand-Target Pair